AKT inhibitor is a broadly selective, potent, ATP-competitive Akt inhibitor, displays 900-fold greater selectivity for PKB (IC50 = 0.5 nM) than PKA (IC50=450 nM).
For research use only. We do not sell to patients.
Name | AKT inhibitor |
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Iupac Chemical Name | N-[[(3S)-3-AMINO-1-(5-ETHYL-7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)-3-PYRROLIDINYL]METHYL]-2,4-DIFLUORO-BENZAMIDE |
Synonyms | AKT inhibitor;AKT protein kinase inhibitor |
Molecular Formula | C20H22F2N6O |
Molecular Weight | 400.43 |
Smile | N[C@]1(CN(CC1)C=1C2=C(N=CN1)NC=C2CC)CNC(C2=C(C=C(C=C2)F)F)=O |
InChiKey | MOZRQQTUYAYCQT-FQEVSTJZSA-N |
InChi | InChI=1S/C20H22F2N6O/c1-2-12-8-24-17-16(12)18(27-11-26-17)28-6-5-20(23,10-28)9-25-19(29)14-4-3-13(21)7-15(14)22/h3-4,7-8,11H,2,5-6,9-10,23H2,1H3,(H,25,29)(H,24,26,27)/t20-/m0/s1 |
CAS Number | 1004990-28-6 |
Related CAS |
Packaging | Price | Availability | Purity | Shipping Time |
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Formulation | crystalline solid |
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Purity | 98% |
Storage | 3 years -20ºCpowder |
Solubility | Soluble in DMSO |
Handling | |
Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. |
HS Code |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |