BAY-1316957 is a highly potent, selective, orally available human prostaglandin E2 receptor subtype 4 (hEP4-R) antagonist (IC50= 15.3 nM ) with excellent drug metabolism and pharmacokinetics properties.
For research use only. We do not sell to patients.
Name | BAY-1316957 |
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Iupac Chemical Name | 2-(9-Ethyl-6-methyl-9H-carbazol-3-yl)-1-(2-methoxyethyl)-4-methyl-1H-benzimidazole-5-carboxylic acid |
Synonyms | BAY-1316957; BAY 1316957; BAY1316957; |
Molecular Formula | C27H27N3O3 |
Molecular Weight | 441.531 |
Smile | O=C(C1=CC=C2C(N=C(C3=CC4=C(C=C3)N(CC)C5=C4C=C(C)C=C5)N2CCOC)=C1C)O |
InChiKey | FHXIZAPGGULPIK-UHFFFAOYSA-N |
InChi | InChI=1S/C27H27N3O3/c1-5-29-22-9-6-16(2)14-20(22)21-15-18(7-10-23(21)29)26-28-25-17(3)19(27(31)32)8-11-24(25)30(26)12-13-33-4/h6-11,14-15H,5,12-13H2,1-4H3,(H,31,32) |
CAS Number | 1613264-40-6 |
Related CAS |
Packaging | Price | Availability | Purity | Shipping Time |
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Bulk | Enquiry | Enquiry | Enquiry |
Formulation | Off-white solid to white solid |
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Purity | >98% |
Storage | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
Solubility | Soluble in DMSO |
Handling | |
Shipping Condition | Shipped under ambient temperature |
HS Code |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |