CP-506 (SN-36506) is an hypoxia-activated prodrug of a DNA-alkylating nitrogen mustard compound capable of selectively targeting tumor cells and designed to have good aqueous solubility, good oral bioavailability and no off-mechanism activation by the human aerobic reductase AKR1C3.
For research use only. We do not sell to patients.
Name | CP-506 ( Synonyms: SN-36506 ) |
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Iupac Chemical Name | Methanesulfonic acid 2-[(2-bromoethyl)[5-(4-ethylpiperazine-1-carbonyl)-2-(methanesulfonyl)-4-nitrophenyl]amino]ethyl methanesulfonate |
Synonyms | CP-506 ; SN-36506 ; CP 506 ; SN 36506 ; CP506 ; SN36506 |
Molecular Formula | C20H33BrN4O11S3 |
Molecular Weight | 681.59 |
Smile | CS(=O)(O)=O.CS(=O)(OCCN(CCBr)C1=CC(C(N2CCN(CC)CC2)=O)=C([N+]([O-])=O)C=C1S(=O)(C)=O)=O |
InChiKey | WJUPXQLICCCCRQ-UHFFFAOYSA-N |
InChi | InChI=1S/C19H29BrN4O8S2.CH4O3S/c1-4-21-7-9-23(10-8-21)19(25)15-13-17(18(33(2,28)29)14-16(15)24(26)27)22(6-5-20)11-12-32-34(3,30)31;1-5(2,3)4/h13-14H,4-12H2,1-3H3;1H3,(H,2,3,4) |
CAS Number | 2227304-19-8 |
Related CAS | 2227304-19-8 |
Packaging | Price | Availability | Purity | Shipping Time |
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Bulk | Enquiry | Enquiry | Enquiry |
Formulation | Solid powder |
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Purity | 98% Min. |
Storage | Dry, dark and at 0 - 4℃ for short term (days to weeks) or -20℃ for long term (months to years). |
Solubility | Soluble in DMSO |
Handling | Refer to MSDS |
Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
HS Code | 2934200090 |
Targets | |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |