DC-S100 is a selective histone methyltransferase SET7 inhibitor.
For research use only. We do not sell to patients.
Name | DC-S100 |
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Iupac Chemical Name | N-(3,4-Dimethoxy-phenyl)-4-nitro-benzamide |
Synonyms | DC-S100; DC S100; DCS100; |
Molecular Formula | C15H14N2O5 |
Molecular Weight | 302.28 |
Smile | O=C(NC1=CC=C(OC)C(OC)=C1)C2=CC=C([N+]([O-])=O)C=C2 |
InChiKey | QVRYMECVJRSTFI-UHFFFAOYSA-N |
InChi | InChI=1S/C15H14N2O5/c1-21-13-8-5-11(9-14(13)22-2)16-15(18)10-3-6-12(7-4-10)17(19)20/h3-9H,1-2H3,(H,16,18) |
CAS Number | 178803-91-3 |
Related CAS |
Packaging | Price | Availability | Purity | Shipping Time |
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Bulk | Enquiry | Enquiry | Enquiry |
Formulation | Solid powder |
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Purity | 98% Min. |
Storage | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
Solubility | Soluble in DMSO |
Handling | |
Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
HS Code |
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Mechanism | |
Cell study | |
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Clinical study |
1: Meng F, Cheng S, Ding H, Liu S, Liu Y, Zhu K, Chen S, Lu J, Xie Y, Li L, Liu R, Shi Z, Zhou Y, Liu YC, Zheng M, Jiang H, Lu W, Liu H, Luo C. Discovery and Optimization of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Pharmacophore- and Docking-Based Virtual Screening. J Med Chem. 2015 Oct 22;58(20):8166-81. doi: 10.1021/acs.jmedchem.5b01154. Epub 2015 Sep 30. PubMed PMID: 26390175.
2: Furihata M, Ohtsuki Y, Ido E, Iwata J, Sonobe H, Araki K, Ogoshi S, Ohmori K. HLA-DR antigen- and S-100 protein-positive dendritic cells in esophageal squamous cell carcinoma--their distribution in relation to prognosis. Virchows Arch B Cell Pathol Incl Mol Pathol. 1992;61(6):409-14. PubMed PMID: 1349780.