Elinzanetant ( NT-814 )
Catalog No: 20259
CAS Number: 929046-33-3
Purity: ≧98.0%
Elinzanetant, previously known as NT-814 (45), is a dual NK1,3R antagonist and therefore has the potential to reduce GnRH pulsatility by blocking the endogenous effects of NKB and SP on the reproductive axis.
For research use only. We do not sell to patients.
Chemical Information
| Name | Elinzanetant ( NT-814 ) |
|---|---|
| Iupac Chemical Name | 2-[3,5-bis(trifluoromethyl)phenyl]-N-{4-(4-fluoro-2-methylphenyl)-6-[(7S,9aS)-7-(hydroxymethyl)hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]pyridin-3-yl}-N,2-dimethylpropanamide |
| Synonyms | Elinzanetant ; GSK1144814A ; NT-814 ; NT 814 ; NT814 ; GSK-1144814A ; GSK 1144814A |
| Molecular Formula | C33H35F7N4O3 |
| Molecular Weight | 668.64 |
| Smile | CC(C)(C1=CC(C(F)(F)F)=CC(C(F)(F)F)=C1)C(N(C2=C(C3=CC=C(F)C=C3C)C=C(N4C[C@@]5([H])COCCN5C[C@H]4CO)N=C2)C)=O |
| InChiKey | DWRIJNIPBUFCQS-DQEYMECFSA-N |
| InChi | InChI=1S/C33H35F7N4O3/c1-19-9-23(34)5-6-26(19)27-13-29(44-16-25-18-47-8-7-43(25)15-24(44)17-45)41-14-28(27)42(4)30(46)31(2,3)20-10-21(32(35,36)37)12-22(11-20)33(38,39)40/h5-6,9-14,24-25,45H,7-8,15-18H2,1-4H3/t24-,25-/m0/s1 |
| CAS Number | 929046-33-3 |
| Related CAS | 929046-33-3 |
Ordering Information
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Off-white Solid |
|---|---|
| Purity | ≧98.0% |
| Storage | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Handling | Avoid inhalation, contact with eyes and skin. Avoid dust and aerosol formation. Use only in areas with appropriate exhaust ventilation. |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| HS Code |
Coming soon.
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |
Not available
Chemical Structure
