Ensifentrine ( RPL554 )
Catalog No: 61726
CAS Number: 1884461-72-6
Purity: ≧98.0%
Ensifentrine (RPL554) is an investigational, first-in-class, inhaled dual inhibitor of PDE 3 and 4 that combines bronchodilator and anti-inflammatory actions in a single compound.
For research use only. We do not sell to patients.
Chemical Information
| Name | Ensifentrine ( RPL554 ) |
|---|---|
| Iupac Chemical Name | N-(2-{(2E)-9,10-dimethoxy-4-oxo-2-[(2,4,6- trimethylphenyl)imino]-6,7-dihydro-2H-pyrimido[6,1- a]isoquinolin-3(4H)-yl}ethyl)urea |
| Synonyms | Ensifentrine ; RPL554 ; RPL-554 ; RPL 554 |
| Molecular Formula | C26H31N5O4 |
| Molecular Weight | 477.565 |
| Smile | O=C(N)NCCN1C(N(CCC2=C3C=C(OC)C(OC)=C2)C3=C/C1=N\C4=C(C)C=C(C)C=C4C)=O |
| InChiKey | CSOBIBXVIYAXFM-BYNJWEBRSA-N |
| InChi | InChI=1S/C26H31N5O4/c1-15-10-16(2)24(17(3)11-15)29-23-14-20-19-13-22(35-5)21(34-4)12-18(19)6-8-30(20)26(33)31(23)9-7-28-25(27)32/h10-14H,6-9H2,1-5H3,(H3,27,28,32)/b29-23+ |
| CAS Number | 1884461-72-6 |
| Related CAS | 1884461-72-6 |
Ordering Information
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | light-yellow solid |
|---|---|
| Purity | ≧98.0% |
| Storage | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Handling | Avoid inhalation, contact with eyes and skin. Avoid dust and aerosol formation. Use only in areas with appropriate exhaust ventilation. |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| HS Code | 2933999701 |
Coming soon.
| Targets | dual phosphodiesterase 3/4 inhibitor |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |
Not available
Chemical Structure
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