GSK269962A
Catalog No: 102206
CAS Number: 850664-21-0
Purity: 98%
GSK269962A(CAS 850664-21-0) is a potent ROCK inhibitor (IC50 values are 1.6 and 4 nM for recombinant human ROCK1 and ROCK2 respectively); displays greater than 30-fold selectivity for ROCK against a panel of serine/threonine kinases.
For research use only. We do not sell to patients.
Chemical Information
| Name | GSK269962A |
|---|---|
| Iupac Chemical Name | N-(3-{[2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-1H-imidazo[4,5-c] pyridin-6-yl]oxy}phenyl)-4-[2-(4-morpholinyl)ethoxy]benzamide |
| Synonyms | GSK 269962A; GSK-269962A; GSK269962; GSK 269962; GSK-269962 |
| Molecular Formula | C29H30N8O5 |
| Molecular Weight | 570.6 |
| Smile | NC=1C(=NON1)C=1N(C2=C(C=NC(=C2)OC=2C=C(C=CC2)NC(C2=CC=C(C=C2)OCCN2CCOCC2)=O)N1)CC |
| InChiKey | YOVNFNXUCOWYSG-UHFFFAOYSA-N |
| InChi | InChI=1S/C29H30N8O5/c1-2-37-24-17-25(31-18-23(24)33-28(37)26-27(30)35-42-34-26)41-22-5-3-4-20(16-22)32-29(38)19-6-8-21(9-7-19)40-15-12-36-10-13-39-14-11-36/h3-9,16-18H,2,10-15H2,1H3,(H2,30,35)(H,32,38) |
| CAS Number | 850664-21-0 |
| Related CAS |
Ordering Information
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Solid powder |
|---|---|
| Purity | 98% |
| Storage | -20 ºC for 3 years |
| Solubility | Soluble in DMSO |
| Handling | |
| Shipping Condition | Shipped under ambient temperature |
| HS Code |
Coming soon.
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |
Not available
Chemical Structure
