GSK3787 is as a selective and irreversible antagonist of PPAR with pIC50 of 6.6, with no measurable affinity for hPPAR or hPPAR.
For research use only. We do not sell to patients.
Name | GSK3787 |
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Iupac Chemical Name | Benzamide, 4-chloro-N-[2-[[5-(trifluoromethyl)-2-pyridinyl]sulfonyl]ethyl]- |
Synonyms | N/A |
Molecular Formula | C15H12ClF3N2O3S |
Molecular Weight | 392.78 |
Smile | ClC1=CC=C(C(=O)NCCS(=O)(=O)C2=NC=C(C=C2)C(F)(F)F)C=C1 |
InChiKey | JFUIMTGOQCQTPF-UHFFFAOYSA-N |
InChi | InChI=1S/C15H12ClF3N2O3S/c16-12-4-1-10(2-5-12)14(22)20-7-8-25(23,24)13-6-3-11(9-21-13)15(17,18)19/h1-6,9H,7-8H2,(H,20,22) |
CAS Number | 188591-46-0 |
Related CAS |
Packaging | Price | Availability | Purity | Shipping Time |
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Bulk | Enquiry | Enquiry | Enquiry |
Formulation | off-white solid |
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Purity | 98% |
Storage | 3 years -20ºCpowder |
Solubility | 2mg/ml in DMSO |
Handling | |
Shipping Condition | Shipped under ambient temperature |
HS Code |
Targets | |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |