KB-0742 is a Potent, Selective, Orally Bioavailable Small Molecule Inhibitor of CDK9 for MYC-Dependent Cancers.
For research use only. We do not sell to patients.
Name | KB-0742 |
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Iupac Chemical Name | (1S,3S)-N3-[5-(1-ethylpropyl)pyrazolo[1,5-a]pyrimidin-7-yl]cyclopentane-1,3-diamine |
Synonyms | KB-0742 ; KB 0742 ; KB0742 |
Molecular Formula | C16H25N5 |
Molecular Weight | 287.41 |
Smile | N[C@@H]1C[C@@H](NC2=CC(C(CC)CC)=NC3=CC=NN23)CC1 |
InChiKey | VYKCLMALANGCDF-STQMWFEESA-N |
InChi | InChI=1S/C16H25N5/c1-3-11(4-2)14-10-16(19-13-6-5-12(17)9-13)21-15(20-14)7-8-18-21/h7-8,10-13,19H,3-6,9,17H2,1-2H3/t12-,13-/m0/s1 |
CAS Number | 2416873-83-9 |
Related CAS | 2416873-83-9 ; 2990122-63-7 |
Packaging | Price | Availability | Purity | Shipping Time |
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Bulk | Enquiry | Enquiry | Enquiry |
Formulation | Off-white solid |
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Purity | ≧98.0% |
Storage | Dry, dark and at 0 - 4℃ for short term (days to weeks) or -20℃ for long term (months to years). |
Solubility | Soluble in DMSO (DMSO : ≥ 100 mg/mL) |
Handling | Refer to MSDS |
Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
HS Code | 2934200090 |
Targets | CDK Inhibitor |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |