Nelotanserin(APD125) is a potent and selective human 5-hydroxytryptamine2A inverse agonist for the treatment of insomnia.
For research use only. We do not sell to patients.
Name | Nelotanserin |
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Iupac Chemical Name | 1-(3-(4-bromo-1-methyl-1H-pyrazol-5-yl)-4-methoxyphenyl)-3-(2,4-difluorophenyl)urea |
Synonyms | APD125; APD-125; Nelotanserin |
Molecular Formula | C18H15BrF2N4O2 |
Molecular Weight | 437.24 |
Smile | O=C(NC1=CC=C(F)C=C1F)NC2=CC=C(OC)C(C3=C(Br)C=NN3C)=C2 |
InChiKey | COSPVUFTLGQDQL-UHFFFAOYSA-N |
InChi | InChI=1S/C18H15BrF2N4O2/c1-25-17(13(19)9-22-25)12-8-11(4-6-16(12)27-2)23-18(26)24-15-5-3-10(20)7-14(15)21/h3-9H,1-2H3,(H2,23,24,26) |
CAS Number | 839713-36-9 |
Related CAS |
Packaging | Price | Availability | Purity | Shipping Time |
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Bulk | Enquiry | Enquiry | Enquiry |
Formulation | Off-white solid to white solid |
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Purity | >98% |
Storage | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
Solubility | Soluble in DMSO, not in water |
Handling | |
Shipping Condition | Shipped under ambient temperature |
HS Code |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |