PZM21 is a potent Gi activator with exceptional selectivity for μOR and minimal β-arrestin-2 recruitment.
For research use only. We do not sell to patients.
Name | PZM21 |
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Iupac Chemical Name | 1-[(2S)-2-(Dimethylamino)-3-(4-hydroxyphenyl)propyl]-3-[(2S)-1-(thiophen-3-yl)propan-2-yl]urea |
Synonyms | PZM21; PZM-21; PZM 21. |
Molecular Formula | C19H27N3O2S |
Molecular Weight | 361.504 |
Smile | O=C(N[C@@H](C)CC1=CSC=C1)NC[C@@H](N(C)C)CC2=CC=C(O)C=C2 |
InChiKey | MEDBIJOVZJEMBI-YOEHRIQHSA-N |
InChi | InChI=1S/C19H27N3O2S/c1-14(10-16-8-9-25-13-16)21-19(24)20-12-17(22(2)3)11-15-4-6-18(23)7-5-15/h4-9,13-14,17,23H,10-12H2,1-3H3,(H2,20,21,24)/t14-,17-/m0/s1 |
CAS Number | 1997387-43-5 |
Related CAS |
Packaging | Price | Availability | Purity | Shipping Time |
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Bulk | Enquiry | Enquiry | Enquiry |
Formulation | Off-white solid to white solid |
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Purity | >98% |
Storage | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
Solubility | Soluble in DMSO |
Handling | |
Shipping Condition | Shipped under ambient temperature |
HS Code |
Targets | |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |