SB-742457(Intepirdine) is a highly selective 5-HT6 receptor antagonist with pKi of 9.63; exhibits >100-fold selectivity over other receptors.
For research use only. We do not sell to patients.
Name | SB-742457 ( Intepirdine ) |
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Iupac Chemical Name | 3-(benzenesulfonyl)-8-piperazin-1-ylquinoline |
Synonyms | GSK-742457 ; RVT-101 ; Intepirdine ; SB-742457 ; SB742457 |
Molecular Formula | C19H19N3O2S |
Molecular Weight | 353.438 |
Smile | C1CN(CCN1)C2=CC=CC3=CC(=CN=C32)S(=O)(=O)C4=CC=CC=C4 |
InChiKey | JJZFWROHYSMCMU-UHFFFAOYSA-N |
InChi | InChI=1S/C19H19N3O2S/c23-25(24,16-6-2-1-3-7-16)17-13-15-5-4-8-18(19(15)21-14-17)22-11-9-20-10-12-22/h1-8,13-14,20H,9-12H2 |
CAS Number | 607742-69-8 |
Related CAS | 607742-69-8 |
Packaging | Price | Availability | Purity | Shipping Time |
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Bulk | Enquiry | Enquiry | Enquiry |
Formulation | Light-yellow solid |
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Purity | 98% |
Storage | -20 ºC for 3 years |
Solubility | Soluble in DMSO |
Handling | Avoid inhalation, contact with eyes and skin. Avoid dust and aerosol formation. Use only in areas with appropriate exhaust ventilation. |
Shipping Condition | Shipped under ambient temperature |
HS Code |
Targets | |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |