Balipodect (TAK 063 ) is a novel PDE10A inhibitor. It has shown high inhibitory activity and selectivity for human recombinant PDE10A2 in vitro; the half-maximal inhibitory concentration was 0.30 nM, and selectivity over other phosphodiesterases (PDEs) was more than 15000-fold.
Balipodect (TAK 063 ), Bulk in stock,
For research use only. We do not sell to patients.
Name | Balipodect ( TAK-063 ) |
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Iupac Chemical Name | 1-(2-fluoro-4-(1H-pyrazol-1-yl)phenyl)-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one |
Synonyms | TAK063 ;TAK 063 ; Balipodect. |
Molecular Formula | C23H17FN6O2 |
Molecular Weight | 428.42 |
Smile | O=C1C(C2=CC=NN2C3=CC=CC=C3)=NN(C4=CC=C(N5N=CC=C5)C=C4F)C=C1OC |
InChiKey | KVHRYLNQDWXAGI-UHFFFAOYSA-N |
InChi | InChI=1S/C23H17FN6O2/c1-32-21-15-29(19-9-8-17(14-18(19)24)28-13-5-11-25-28)27-22(23(21)31)20-10-12-26-30(20)16-6-3-2-4-7-16/h2-15H,1H3 |
CAS Number | 1238697-26-1 |
Related CAS | 1238697-26-1 |
Packaging | Price | Availability | Purity | Shipping Time |
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Bulk | Enquiry | Enquiry | Enquiry |
Formulation | Light-yellow powder |
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Purity | 98% |
Storage | -20 ºC for 3 years |
Solubility | Soluble in DMSO |
Handling | |
Shipping Condition | Shipped under ambient temperature |
HS Code |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |