TGR-1202 hydrochloride is an orally available, next generation PI3Kdelta inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 and 24.3 nM respectively.
For research use only. We do not sell to patients.
Name | TGR-1202 hydrochloride |
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Iupac Chemical Name | TGR-1202 hydrochloride |
Synonyms | RP5264 hydrochloride; TGR1202 hydrochloride; TGR 1202 hydrochloride; RP-5264 hydrochloride; RP 5264 hydrochloride |
Molecular Formula | C31H25ClF3N5O3 |
Molecular Weight | 608.01 |
InChiKey | |
InChi | |
CAS Number | 1532533-78-0 |
Related CAS |
Packaging | Price | Availability | Purity | Shipping Time |
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Formulation | crystalline solid |
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Purity | 98% |
Storage | 3 years -20℃powder |
Solubility | Soluble in DMSO |
Handling | |
Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |