YCT529, an RAR-α inhibitor, is used as a contraceptive, with a 99% effectiveness. YCT529 acts as a potent and selective antagonist of the Vitamin A receptor retinoic acid receptor alpha (RAR-α). In studies on mice it produced a 99% reduction in sperm production, and it has proceeded to early stage human clinical trials as a potential male contraceptive.
For research use only. We do not sell to patients.
Name | YCT529 |
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Iupac Chemical Name | sodium 4-(5-(2,2-dimethyl-4-(p-tolyl)-2H-chromen-6-yl)-1H-pyrrol-2-yl)benzoate |
Synonyms | YCT529; YCT 529; YCT-529 |
Molecular Formula | C29H24NNaO3 |
Molecular Weight | 457.50 |
Smile | O=C([O-])C1=CC=C(C2=CC=C(C3=CC(C(C4=CC=C(C)C=C4)=CC(C)(C)O5)=C5C=C3)N2)C=C1.[Na+] |
InChiKey | NNFWFHLHNJSJTH-UHFFFAOYSA-M |
InChi | InChI=1S/C29H25NO3.Na/c1-18-4-6-19(7-5-18)24-17-29(2,3)33-27-15-12-22(16-23(24)27)26-14-13-25(30-26)20-8-10-21(11-9-20)28(31)32;/h4-17,30H,1-3H3,(H,31,32);/q;+1/p-1 |
CAS Number | 2863670-67-9 |
Related CAS |
Packaging | Price | Availability | Purity | Shipping Time |
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Bulk | Enquiry | Enquiry | Enquiry |
Formulation | Off-white solid |
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Purity | 98% Min. |
Storage | Dry, dark and at 0 - 4℃ for short term (days to weeks) or -20℃ for long term (months to years). |
Solubility | Soluble in DMSO |
Handling | |
Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
HS Code |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |