Lemborexant(CAS 1369764-02-2)is a novel investigational small molecule that inhibits orexin signaling by binding competitively to both orexin receptor subtypes (orexin receptor 1 and 2).
Lemborexant (E-2006), Bulk in stock, contact us by email for the quotation. Kg scale intermediates are also be provided by custom synthesis.
仅供研究使用。 我们不向患者出售。
名称 | Lemborexant (E-2006) |
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Iupac 化学名称 | (1R,2S)-2-(((2,4-dimethylpyrimidin-5-yl)oxy)methyl)-2-(3-fluorophenyl)-N-(5-fluoropyridin-2-yl)cyclopropanecarboxamide |
同义词 | E-2006; E 2006; E2006; Lemborexant ; Dayvigo |
英文同义词 | E-2006; E 2006; E2006; Lemborexant ; Dayvigo |
分子式 | C22H20F2N4O2 |
分子量 | 410.1554 |
Smile | FC1=CC=CC([C@@]2(COC3=CN=C(C)N=C3C)[C@H](C(NC4=CC=C(F)C=N4)=O)C2)=C1 |
InChiKey | MUGXRYIUWFITCP-PGRDOPGGSA-N |
InChi | InChI=1S/C22H20F2N4O2/c1-13-19(11-25-14(2)27-13)30-12-22(15-4-3-5-16(23)8-15)9-18(22)21(29)28-20-7-6-17(24)10-26-20/h3-8,10-11,18H,9,12H2,1-2H3,(H,26,28,29)/t18-,22+/m0/s1 |
Cas号 | 1369764-02-2 |
相关CAS号 |
包装 | 价格 | 库存 | 纯度 | 备货期 |
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大货 | 询价 | 询价 | 询价 |
外观性状 | Off-white solid |
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纯度 | 98% Min. |
存储 | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
可溶性 | Soluble in DMSO, not in water |
处理方式 | |
运输条件 | Shipped under ambient temperature |
海关编码 |
Targets | |
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Mechanism | |
Cell study | |
Animal study | |
Clinical study |