Balipodect (TAK 063 ) is a novel PDE10A inhibitor. It has shown high inhibitory activity and selectivity for human recombinant PDE10A2 in vitro; the half-maximal inhibitory concentration was 0.30 nM, and selectivity over other phosphodiesterases (PDEs) was more than 15000-fold.
Balipodect (TAK 063 ), Bulk in stock,
仅供研究使用。 我们不向患者出售。
名称 | Balipodect ( TAK-063 ) |
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Iupac 化学名称 | 1-(2-fluoro-4-(1H-pyrazol-1-yl)phenyl)-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one |
同义词 | TAK063 ; TAK 063 ; Balipodect. |
英文同义词 | TAK063 ;TAK 063 ; Balipodect. |
分子式 | C23H17FN6O2 |
分子量 | 428.42 |
Smile | O=C1C(C2=CC=NN2C3=CC=CC=C3)=NN(C4=CC=C(N5N=CC=C5)C=C4F)C=C1OC |
InChiKey | KVHRYLNQDWXAGI-UHFFFAOYSA-N |
InChi | InChI=1S/C23H17FN6O2/c1-32-21-15-29(19-9-8-17(14-18(19)24)28-13-5-11-25-28)27-22(23(21)31)20-10-12-26-30(20)16-6-3-2-4-7-16/h2-15H,1H3 |
Cas号 | 1238697-26-1 |
相关CAS号 | 1238697-26-1 |
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