TGR5 Receptor Agonist, a potent TGR5(GPCR19) agonist, showed improved potency in the U2-OS cell assay (pEC50 = 6.8) and in melanophore cells (pEC50 = 7.5).
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化学信息
名称 | TGR5 Receptor Agonist |
分子式 | C18H14Cl2N2O2 |
分子量 | 361.22 |
Smile | Cc1c(c(no1)c2ccccc2Cl)C(=O)N(C)c3ccc(cc3)Cl |
InChiKey | IGRCWJPBLWGNPX-UHFFFAOYSA-N |
InChi | InChI=1S/C18H14Cl2N2O2/c1-11-16(17(21-24-11)14-5-3-4-6-15(14)20)18(23)22(2)13-9-7-12(19)8-10-13/h3-10H,1-2H3 |
Cas号 | 1197300-24-5 |
MDL | MFCD17169972 |
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