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CDK

编号化学名称Cas号纯度
52105SNS-032 ( BMS-387032 )
SNS-032 has firstly been described as a selective inhibitor ofCDK2withIC50of 48 nM an
345627-80-798% 
51614AMG-925
AMG-925 is a potent and orally bioavailable dual inhibitor of CDK4 and FLT3, includin
1401033-86-098% 
2073106Lerociclib HCl (G1T38 HCl)
Lerociclib HCl (G1T38 dihydrochloride)是一种分化型口服CDK4 / 6抑制剂,对
2097938-59-3≧98.0%
185235Trilaciclib (G1T28)
Trilaciclib是一种小分子竞争性细胞周期蛋白依赖性激酶4和6(CDK4 /
1374743-00-6>98%
204302Lerociclib
Lerociclib,也称为G1T38,是一种口服,有效和选择性的CDK4 / 6抑制剂
1628256-23-4 (free base)98%
204305ICEC0942 HCl
ICEC0942, also known as PPDA-001 and CT7001, is a potent, orally active and selective
1805789-54-1 (HCl)98% Min.
2073107Trilaciclib hydrochloride (G1T28 hydrochloride)
Trilaciclib是一种小分子竞争性细胞周期蛋白依赖性激酶4和6(CDK4 /
1977495-97-898% Min.
62502TG02 ( SB1317 )
SB1317 (TG02) is a novel small molecule potent CDK/JAK2/FLT3 inhibitor. SB1317 was so
937270-47-8≧98.0%
236271TP1287
Alvocidib Prodrug TP-1287 is an orally bioavailable, highly soluble phosphate prodrug
2044686-42-0≧97.0%
237071Flavopiridol ( 夫拉平度 )
Alvocidib is a synthetic dihydroxyflavone that is 5,7-dihydroxyflavone which is subst
146426-40-6≧98.0%