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抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
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订购信息
联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
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产品名字索引 H
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产品名字索引 H
HFY-4A
(Catalog# : 20661, Cas# :
2094810-82-7
)
HFY-4A is a HDAC inhibitor. HFY-4A inhibits breast cancer cell proliferation, migrati
Hynic-TOC
(Catalog# : 20658, Cas# :
257943-19-4
)
Hynic-TOC is a ligand for making 99mTc-Hynic-TOC as an imaging agent in the diagnosti
HDAC-IN-58
(Catalog# : 20568, Cas# :
2071224-39-8
)
HDAC-IN-58 is a HDAC inhibitor.
4,5-二碘-1H-1H-1,2,3-三氮唑
(Catalog# : 20521, Cas# :
28194-09-4
)
HM43239
(Catalog# : 20517, Cas# :
2569527-64-4
)
HM43239 is an orally active small molecule inhibitor of FLT3 that selectively inhibit
5-溴-6-环丙基嘧啶-4-醇
(Catalog# : 20482, Cas# :
27192-20-7
)
2(1H)-Pyridinone, 5,6-dihydro-4-(4-methylphenyl)-3-(2H-tetrazol-5-yl)-6-[4-(4,4,4-trifluorobutoxy)phenyl]-6-(trifluoromethyl)-, (6S)-
(Catalog# : 20430, Cas# :
1441057-15-3
)
1H-Indazole-1-acetic acid, 3-acetyl-5-bromo-, 1,1-dimethylethyl ester
(Catalog# : 20422, Cas# :
2086183-72-2
)
4-氯-1-[三(甲基乙基)硅酯]-1H-吡咯并[2,3-B]吡啶
(Catalog# : 20410, Cas# :
651744-48-8
)
4-hydroxybiphenyl-4-carboxamide
(Catalog# : 20404, Cas# :
182318-78-1
)
1H-吡咯并[2,3-B]吡啶-2-羧酸乙酯
(Catalog# : 20388, Cas# :
221675-35-0
)
6-羟基-3,4-二氢-1H-2-萘酮
(Catalog# : 20371, Cas# :
52727-28-3
)
HISPOLON(P)
(Catalog# : 210201, Cas# :
173933-40-9
)
HMPL-523
(Catalog# : 20123101, Cas# :
1415792-84-5
)
HMPL-523 is a novel, highly selective and potent small molecule oral inhibitor target
5-Hydroxymethyldeoxyuridine
(Catalog# : 2091910, Cas# :
5116-24-5
)
5-Hydroxymethyldeoxyuridine is a nucleoside analog with anticancer and antiviral acti
2,4-二甲基-5-羟基嘧啶
(Catalog# : 2091204, Cas# :
412003-95-3
)
我们可以生产公斤级的2,4-二甲基-5-羟基嘧啶 (CAS 412003-95-3)。
H-BETA-ALA-AMC TFA
(Catalog# : 2071633, Cas# :
201847-54-3
)
2'-HYDROXY-6'-METHOXYACETOPHENONE
(Catalog# : 2062006, Cas# :
703-23-1
)
HC-070
(Catalog# : 206104, Cas# :
1628291-95-1
)
HC-070 is a potent inhibitor of TRPC4 and TRPC5, leading to anxiolytic and antidepres
Hydroxyfasudil HCl
(Catalog# : 204610, Cas# :
155558-32-0 (HCl)
)
Hydroxyfasudil, aslo known as HA1100, is a cell-permeable hydroxylated metabolite of
HBX-41108
(Catalog# : 19317, Cas# :
924296-39-9
)
HBX 41108是泛素特异性蛋白酶(USP) 7的抑制剂。HBX 41108通过IC(50)在亚
HS-1371
(Catalog# : 192223, Cas# :
2158197-70-5
)
HS-1371是一种新型的RIP3-介导坏死性凋亡激酶抑制剂。HS-1371以ATP-竞
HZ-1157
(Catalog# : 19182, Cas# :
1009734-33-1
)
HZ-1157是一种丙肝病毒(HCV)抑制剂,对HCV NS3/4A蛋白酶有抑制作用。
H 151
(Catalog# : 1811022, Cas# :
941987-60-6
)
H 151是一种诱捕拮抗剂,共价结合在Cys91上,阻断棕榈酰化和防止
HC-056456
(Catalog# : 1810171, Cas# :
7733-96-2
)
HC-056456是CatSper的通道调制器。
20-HETE
(Catalog# : 185283, Cas# :
79551-86-3
)
20-HETE是一种细胞色素P450 (CYP450)代谢产物,在脑血管和肾血管中扮
HMN-154
(Catalog# : 184122, Cas# :
173528-92-2
)
HMN-154是一种苯磺胺的抗癌剂。HMN-154通过剂量依赖性的方式抑制NF
HJC0152
(Catalog# : 1710133, Cas# :
1420290-99-8
)
HJC0152是对人的头部和颈部鳞状细胞癌(鳞癌)的信号转导与转录
9-Hydroxyellipticin(free base)
(Catalog# : 1791313, Cas# :
51131-85-2
)
9-hydroxyellipticine,又名 IGIG 929和LS133324,是一种强效的细胞毒和抗
H3B-6527
(Catalog# : 179822, Cas# :
1702259-66-2
)
H3B-6527是一个强有力的口服活性分子抑制剂,具有潜在的抗肿瘤活
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
PLX8394
(Catalog# : 20613, Cas# :
1393466-87-9
)
PLX8394 is an orally bioavailable inhibitor of serine/threonine-protein kinase B-raf
Zelasudil
(Catalog# : 24014, Cas# :
2365193-22-0
)
Zelasudil 是一种有效的、高选择性的口服活性抑制剂,针对 Rho 相关
Ziftomenib ( KO-539 )
(Catalog# : 24013, Cas# :
2134675-36-6
)
Ziftomenib 是一种口服、有效、选择性的小分子抑制剂,针对 menin 和
Zunsemetinib
(Catalog# : 24012, Cas# :
1640282-42-3
)
Zunsemetinib是一种在研口服丝裂原活化蛋白激酶活化蛋白激酶2(MK2
Zongertinib ( BI 1810631 )
(Catalog# : 24011, Cas# :
2728667-27-2
)
Zongertinib [BI 1810631] 是一种人表皮生长因子受体 2 (HER2) 抑制剂。
Zasocitinib
(Catalog# : 24010, Cas# :
2272904-53-5
)
Zasocitinib是一种作用于非受体酪氨酸蛋白激酶 (TYK2)靶点的抑制
RNK-05047
(Catalog# : 24008, Cas# :
2503036-46-0
)
RNK-05047 为BRD4降解剂,其在小鼠荷瘤异种移植模型中展现出显著抑
Asengeprast (FT011)
(Catalog# : 24009, Cas# :
1001288-58-9
)
Asengeprast (FT011) 是一种抗纤维化剂,降低胶原蛋白 I 和 III 的 mRNA
ERAS-801 ( JGK-068S )
(Catalog# : 20635, Cas# :
2490431-16-6
)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。
T-1095
(Catalog# : 24004, Cas# :
209746-59-8
)
T-1095 is a potent and selective inhibitor of Na+-glucose cotransporters (SGLTs).