武汉永璨生物科技有限公司
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抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
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MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
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Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
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others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
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Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
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订购信息
联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
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订购信息
联系我们
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联系我们
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产品名字索引 R
Remetinostat
(Catalog# : 193111, Cas# :
946150-57-8
)
Remetinostat,也被称为SHP-141,是一种外用制剂,含有组蛋白脱乙酰
RG7834
(Catalog# : 19355, Cas# :
2072057-17-9
)
RG7834,也称为RO7020322,是一种新型口服HBV病毒基因表达抑制剂阻断病
RWJ-56110
(Catalog# : 19353, Cas# :
252889-88-6
)
RWJ-56110是一种选择性蛋白酶活化受体-1 (PAR1)拮抗剂。它阻断凝血酶
RBC8
(Catalog# : 19313, Cas# :
361185-42-4
)
RBC8是一种RalA和RalB GTPase抑制剂(EC50 ~ 3.5μM)。RBC8抑制小鼠异种移植
Rogaratinib
(Catalog# : 192277, Cas# :
1443530-05-9
)
Rogaratinib, 也称为BAY-1163877, 是一种异常的成纤维细胞生长因子受体
Rebimastat
(Catalog# : 192254, Cas# :
259188-38-0
)
Rebimastat,又名BMS275291,是一种具有潜在抗肿瘤活性的巯基第二代
Retosiban
(Catalog# : 192193, Cas# :
820957-38-8
)
Retosiban,又称GSK-221149-A;是一种口服活性强、选择性强的亚纳米(Ki
RKI-1313
(Catalog# : 19183, Cas# :
1342276-76-9
)
RKI-1313是RKI-1447 (GLXC-05200)的阴性对照,是Rho-相关ROCK激酶的有效抑
RGX-104 free form
(Catalog# : 19181, Cas# :
610318-54-2
)
RGX-104,又称SB 742881,是肝脏X受体激动剂,具有潜在的免疫调节和
R547
(Catalog# : 1811151, Cas# :
741713-40-6
)
R547是口服生物有效的二氨基嘧啶环磷酰胺依赖性激酶抑制剂(CDKI)
Regadenoson
(Catalog# : 1810224, Cas# :
313348-27-5
)
Regadenoson是一种A2A腺苷受体激动剂,是一种冠状血管舒张剂,通常
Resminostat
(Catalog# : 18751, Cas# :
864814-88-0
)
Resminostat,又称4S-201和RAS2410,是一种口服生物可获得的组蛋白去乙
RMC-4550
(Catalog# : 186251, Cas# :
2172651-73-7
)
RMC-4550一种有效且具有选择性的SHP2抑制剂。
RGX-104盐酸盐
(Catalog# : 186234, Cas# :
610318-03-1
)
RGX-104是一种具有潜在免疫调节和抗肿瘤活性的肝X受体激动剂。
Resminostat HCl
(Catalog# : 185317, Cas# :
1187075-34-8
)
Resminostat HCl是一种有效的HDAC1/3/6抑制剂。
Rovazolac
(Catalog# : 185234, Cas# :
1454288-88-0
)
Rovazolac是一种抗炎药。
Rolapitant游离
(Catalog# : 185152, Cas# :
5552292-08-7
)
Rolapitant,也被称为SCH-619734,是一种口服生物可用的,具有中央作
RO10-5824
(Catalog# : 185141, Cas# :
189744-46-5
)
RO10-5824是一种D4-选择性局部激动剂。RO10-5824是管理可卡因使用障碍
利卡司琼
(Catalog# : 184281, Cas# :
117086-68-7
)
利卡司琼,也称为Brl 46470,是止吐剂。
R-IMPP
(Catalog# : 18413, Cas# :
2133832-83-2
)
R-IMPP是PCSK9的转化抑制剂。
Rimegepant
(Catalog# : 18441, Cas# :
1289023-67-1
)
Rimegepant,也称为BMS-927711,在治疗偏头痛的临床试验中,是一种有
Ritlecitinib ( PF-06651600 )
(Catalog# : 18435, Cas# :
1792180-81-4
)
Ritlecitinib ( PF-06651600 )是一种有效的选择性JAK3抑制剂,是一种具有
R-GNE-140
(Catalog# : 18432, Cas# :
2003234-63-5
)
R-GNE-140是一种新型高效的乳酸脱氢酶(LDHA)抑制剂,LDHA的IC50为3nM,
(2R,14R)-4-((R)-1-((R)-4-benzyl-2-oxooxazolidin-3-yl)-3-(tert-butoxycarbonyl)-1-oxopropan-2-yl)benzyl 2,4-dimethylbenzoate
(Catalog# : 183217, Cas# :
2097334-19-3
)
(2R,14R)-4-((R)-1-((R)-4-benzyl-2-oxooxazolidin-3-yl)-3-(tert-butoxycarbonyl)-1-oxopr
(R)-4-(2-(4-benzyl-2-oxooxazolidin-3-yl)-2-oxoethyl)benzyl 2,4-dimethylbenzoate
(Catalog# : 183216, Cas# :
2097334-18-2
)
(R)-4-(2-(4-benzyl-2-oxooxazolidin-3-yl)-2-oxoethyl)benzyl 2,4-dimethylbenzoate是一
Relebactam
(Catalog# : 1712156, Cas# :
1174018-99-5
)
Relebactam, also known as MK-7655, a potent and selective β-lactamase inhibitor.
盐酸利莫那班
(Catalog# : 179137, Cas# :
158681-13-1
)
利莫那班,又名SR141716,是一种抑制食欲的减肥药。它是为大麻素
Riviciclib HCl
(Catalog# : 179131, Cas# :
920113-03-7
)
Riviciclib,也称为P276-00,是具有潜在抗肿瘤活性的黄酮和细胞周期
RVT-501
(Catalog# : 17917, Cas# :
947620-48-6
)
RVT-501也称为E-6005,是4型磷酸二酯酶(PDE-4)抑制剂用于治疗特应
Roluperidone ( CYR-101 )
(Catalog# : 2017889, Cas# :
359625-79-9
)
Roluperidone, also known as MIN-101, CYR-101, and MT-210, is a 5-HT2A and sigma 2 rec
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
PLX8394
(Catalog# : 20613, Cas# :
1393466-87-9
)
PLX8394 is an orally bioavailable inhibitor of serine/threonine-protein kinase B-raf
Zelasudil
(Catalog# : 24014, Cas# :
2365193-22-0
)
Zelasudil 是一种有效的、高选择性的口服活性抑制剂,针对 Rho 相关
Ziftomenib ( KO-539 )
(Catalog# : 24013, Cas# :
2134675-36-6
)
Ziftomenib 是一种口服、有效、选择性的小分子抑制剂,针对 menin 和
Zunsemetinib
(Catalog# : 24012, Cas# :
1640282-42-3
)
Zunsemetinib是一种在研口服丝裂原活化蛋白激酶活化蛋白激酶2(MK2
Zongertinib ( BI 1810631 )
(Catalog# : 24011, Cas# :
2728667-27-2
)
Zongertinib [BI 1810631] 是一种人表皮生长因子受体 2 (HER2) 抑制剂。
Zasocitinib
(Catalog# : 24010, Cas# :
2272904-53-5
)
Zasocitinib是一种作用于非受体酪氨酸蛋白激酶 (TYK2)靶点的抑制
RNK-05047
(Catalog# : 24008, Cas# :
2503036-46-0
)
RNK-05047 为BRD4降解剂,其在小鼠荷瘤异种移植模型中展现出显著抑
Asengeprast (FT011)
(Catalog# : 24009, Cas# :
1001288-58-9
)
Asengeprast (FT011) 是一种抗纤维化剂,降低胶原蛋白 I 和 III 的 mRNA
ERAS-801 ( JGK-068S )
(Catalog# : 20635, Cas# :
2490431-16-6
)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。
T-1095
(Catalog# : 24004, Cas# :
209746-59-8
)
T-1095 is a potent and selective inhibitor of Na+-glucose cotransporters (SGLTs).