产品目录
| 编号 | 化学名称 | Cas号 | 纯度 | 化学结构 |
|---|---|---|---|---|
| 52026 | AMG-319 | 1608125-21-8 | 98% |  |
| AMG 319 is an investigational, highly selective, small molecule inhibitor of PI3K tha | ||||
| 51614 | AMG-925 | 1401033-86-0 | 98% |  |
| AMG-925 is a potent and orally bioavailable dual inhibitor of CDK4 and FLT3, includin | ||||
| 52640 | ABT-737 | 852808-04-9 | 98% |  |
| ABT-737 is a BH3 mimetic inhibitor ofBcl-xL,Bcl-2andBcl-wwithEC50of 78.7 nM, 30.3 nM | ||||
| 52638 | AZD-7762 | 860352-01-8 | 98% |  |
| AZD7762 is a potent and selective inhibitor of Chk1 with IC50 of 5 nM; equally potent | ||||
| 52626 | AZD1080 | 612487-72-6 | 98% |  |
| AZD1080 is a selective, orally active, brain permeable GSK3 inhibitor of GSK3 and GSK | ||||
| 52617 | A-674563 | 552325-73-2 | 98% |  |
| A-674563 is a potent selective Akt1 inhibitor with an IC50 of 14 nM; also shows inhib | ||||
| 52587 | Alisertib(MLN8237) | 1028486-01-2 | 98% | -cas-1028486-01-2.png) |
| Alisertib (MLN8237) is a selective Aurora A inhibitor with IC50 of 1.2 nM; has >20 | ||||
| 52585 | AMG-208 | 1002304-34-8 | 98% |  |
| AMG-208 is a potent small molecular c-Met inhibitor with an IC50 of 9.3 nM. | ||||
| 52577 | AZD-5438 | 602306-29-6 | 98% |  |
| AZD5438 is a potent inhibitor of CDK1/2/9 with IC50 of 16 nM/6 nM/20 nM. It is less p | ||||
| 52573 | AZD1283 | 919351-41-0 | 98% | |
| AZD1283 is a potent antagonist of the P2Y12 receptor with EC50 of 3.0 ug/kg/min, TI & | ||||
| 52551 | Apoptosis Activator 2 | 79183-19-0 | 98% |  |
| Apoptosis Activator 2 is a potent apoptosis activator; increases procaspase-9 process | ||||
| 52547 | AGI-6780 | 1432660-47-3 | 98% | |
| AGI-6780 is the first highly potent and selective small molecule inhibitor of isocitr | ||||
| 52538 | AP-III-a4 | 1177827-73-4 | 98% | |
| ENOblock(AP-III-a4) is a novel small molecule which is the first, nonsubstrate analog | ||||
| 52533 | AWD 131-138 | 188116-07-6 | 98% |  |
| AWD 131-138(Imepitoin) is a new low-affinity partial benzodiazepine receptor agonist | ||||
| 52524 | Ampalex | 154235-83-3 | 98% |  |
| Ampalex (Ampakine CX516; CX516; BDP 12) is an ampakine and nootropic that acts as an | ||||
| 52523 | AR-A014418 | 487021-52-3 | 98% |  |
| AR-A014418 is a selective and effective GSK3 inhibitor with an IC 50 value of 104 +/- | ||||
| 52504 | AG 18 | 118409-57-7 | 98% |  |
| AG-18(RG-50810; Tyrphostin A23) inhibits EGFR with IC50 of 40 M. | ||||
| 52222 | AG-1478 | 153436-53-4 | 98% |  |
| AG-1478 (NSC 693255) is a selective EGFR inhibitor with IC50 of 3 nM; almost no activ | ||||
| 52240 | Atglistatinc | 1469924-27-3 | 98% |  |
| Atglistatin is a highly potent, selective and competitive inhibitor of adipose trigly | ||||
| 52232 | ATB-346 | 1226895-20-0 | 98% |  |
| ATB-346 is a novel hydrogen sulphide-releasing derivative of naproxen with markedly r | ||||
| 52242 | Afobazole | 173352-21-1 | 98% |  |
| Afobazole (CM346) is an anxiolytic drug; produces anxiolytic and neuroprotective effe | ||||
| 52314 | AT7519 | 844442-38-2 | 98% |  |
| AT7519 is a multi-CDKinhibitor for CDK1, 2, 4, 6 and 9 withIC50of 10-210 nM. It is le | ||||
| 51914 | Aceclofenac | 89796-99-6 | 98% |  |
| Aceclofenac is a non-steroidal anti-inflammatory drug (NSAID) analog of Diclofenac. | ||||
| 51907 | Alectinib(CH5424802) | 1256580-46-7 | 98.5% | -cas-1256580-46-7.png) |
| Alectinibis a second-generation, orally active, potent and highly selective inhibitor | ||||
| 51904 | AZD1152-HQPA | 722544-51-6 | 98% |  |
| Barasertib (AZD1152-HQPA) is a highly selectiveAurora Binhibitor withIC50of 0.37 nM, | ||||
| 51603 | AZD6482 | 1173900-33-8 | ≧98.0% |  |
| AZD6482 is aPI3Kinhibitor withIC50of 10 nM, 8-, 87- and 109-fold more selective to PI | ||||
| 51702 | AZD1208 | 1204144-28-4 | 98% |  |
| AZD1208 is a potent, highly selective, and orally available Pim kinase inhibitor that | ||||
| 51903 | AZ3146 | 1124329-14-1 | 98% |  |
| AZ3146 is a selectiveMps1inhibitor withIC50of ~35 nM, contributes to recruitment of C | ||||
| 51902 | AT13148 | 1056901-62-2 | ≧98% |  |
| AT13148, a first-in-class multi-AGC kinase inhibitor, against gastric cancer cells. A | ||||