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Deuterated
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
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Immunology & Inflammation
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others
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Anilines
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Cas号索引 1
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Cas号索引 1
1240299-33-5 | AZD-3514
(Catalog# : 1810251)
AZD-3514是一种具有潜在抗癌活性的雄激素受体下调因子。
1698055-85-4 | ARS-1620
(Catalog# : 1810222)
ARS-1620是一种具有理想药代动力学的阿托品选择性KRAS-G12C抑制剂。
1175526-27-8 | AM211
(Catalog# : 1810173)
AM-211是前列腺素D2受体2型的一种新型强效拮抗剂。
1190217-35-6 | ASP7663
(Catalog# : 187123)
ASP7663是口服生物可利用选择性TRPA1激活剂。
1188890-28-9 | ABT 702盐酸盐
(Catalog# : 18791)
ABT 702二盐酸盐是一种强效的非核苷腺苷激酶抑制剂,对腺甘酸相
1346623-17-3 | Avacopan
(Catalog# : 18761)
Avacopan也被称为CCX168,是一种口服活性、选择性和有效的C5aR抑制剂
133550-35-3 | AG-494
(Catalog# : 186273)
AG-494,也被称为Tyrphostin AG- 494,是表皮生长因子受体激酶的抑制剂
1869912-39-9 | AZD5153
(Catalog# : 186254)
AZD5153是一种有效的双价三唑吡啶溴化和外治(BET)抑制剂。
1818885-28-7 | ARV-825
(Catalog# : 185253)
ARV-825是一种保护蛋白(蛋白酶-靶向嵌合体)。ARV-825与溴域抑制剂(B
1637771-14-2 | Alobresib
(Catalog# : 185222)
Alobresib是抗肿瘤药物的候选药物。
1467013-03-3 | Adavivint
(Catalog# : 185221)
Adavivint是一种Wnt通道抑制剂和免疫调制剂药物候选者。
1889279-16-6 | A-485
(Catalog# : 185211)
A-485是一种有效且具有选择性的p300/CBP在体外的HAT抑制剂。
1883727-34-1 | AMG-176
(Catalog# : 185185)
AMG-176是诱导髓系白血病细胞分化蛋白MCL-1(骨髓细胞白血病-1)的抑
1217201-17-6 | A-350619盐酸盐
(Catalog# : 185183)
A-350619盐酸盐是可溶性的胍基环酶(sGC)的激活剂。
1253573-53-3 | AMG-511
(Catalog# : 18542)
AMG-511是一种有效的选择性的泛型I PI3K抑制剂。
1186206-79-0 | ALW-II-41-27
(Catalog# : 1842813)
ALW-II-41-27是一种Eph受体酪氨酸激酶抑制剂。
1321514-06-0 | AZD4635
(Catalog# : 184289)
AZD-4635,也叫HTL-1071,是一种口服的小分子腺苷A2A受体拮抗剂。
1229453-99-9 | Acrizanib
(Catalog# : 184181)
Acrizanib,又名LHA510,是一种有效的选择性血管生成抑制剂和VEGFR -
1032570-98-1 | 2-amino-3-methoxy-4-(3-morpholin-4-ylpropoxy)benzonitrile
(Catalog# : 184163)
2-amino-3-methoxy-4-(3-morpholin-4-ylpropoxy)benzonitrile是一种药物中间体。
1058156-90-3 | 安罗替尼
(Catalog# : 184132)
安罗替尼,又名AL3818,是一种受体酪氨酸激酶(RTK)抑制剂,具有潜
1125758-85-1 | A-804598
(Catalog# : 184125)
A-804598是一种P2X7选择性、竞争性的拮抗剂。
185991-07-5 | AMD3465 HCl salt
(Catalog# : 184310)
AMD3465是一种新型CXCR4受体拮抗剂,具有潜在的抗癌和抗艾滋病活性
1220646-23-0 | AVN-492
(Catalog# : 18425)
AVN-492是一种有效且具有选择性的5-HT6R拮抗剂。AVN-492具有良好的体
1173154-32-9 | ALB-127158A
(Catalog# : 18424)
ALB-127158A, also known as ALB-127158(a), is a MCH1 antagonist for the treatment of o
1492952-76-7 | Asciminib ( ABL001 )
(Catalog# : 1711222)
Asciminib, 也叫ABL001,是一种有效的BCR-ABL的变构抑制剂。ABL001在与尼
1644443-47-9 | Autophinib
(Catalog# : 17101617)
Autophinib是一种新颖有效的自噬抑制剂,抑制通过靶向脂质激酶VPS
1124197-79-0 | Adarigiline
(Catalog# : 1710167)
adarigiline是单胺氧化酶B抑制剂的候选药物。
1613589-09-5 | Adafosbuvir
(Catalog# : 1710166)
Adafosbuvir是一种抗病毒药物。
1869912-40-2 | AZD-5153 HNT salt
(Catalog# : 1710161)
AZD-5153 HNT盐,是AZD-5153的6-hydroxy-2-naphthoic酸盐。AZD-5153对抗血液系
1675-66-7 | 阿地米屈
(Catalog# : 179151)
阿地米屈是壬二酸的合成酰胺衍生物,具有对称的化学结构。它被
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
-- PROTAC
----
Molecular Glues
--
Antibody-drug Conjugate/ADC Related
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2991818-13-2 | MGD-28
(Catalog# : 25073)
MGD-28 is a potent molecular glue degrader that demonstrates significant in vitro eff
| TG101209 analog 1
(Catalog# : 25072)
TG101209 analog 1 (Compound 8h) is an inhibitor of BUB1B with an IC50 of 10.36 μ M.
2170729-29-8 | AT-007
(Catalog# : 25071)
AT-007 is an orally active central nervous system (CNS) penetrant Aldose Reductase in
1358751-06-0 | TAK-653
(Catalog# : 25070)
TAK-653 is a novel AMPA receptor potentiator, strictly potentiating a glutamate-induc
1801344-14-8 | Emavusertib
(Catalog# : 25069)
Emavusertib, also known as CA-4948 is a potent IRAK4/FLT3 inhibitor with anti-tumor a
1305267-37-1 | Roginolisib
(Catalog# : 25068)
Roginolisib, also known as MSC2360844 and IOA-244, is a potent, orally active and sel
1198078-60-2 | NT219
(Catalog# : 25067)
NT219 is a novel inhibitor of the insulin/igf signaling cascade (iis), mediating a lo
858128-57-1 | SPB linker
(Catalog# : 25066)
SPB is a agent-linker conjugate for ADC with potent anti-inflammatory activity by usi
1404380-58-0 | JTE-151
(Catalog# : 20594)
JTE-151 是一种 RORγ 抑制剂,可通过抑制与 Th17 细胞活化相关的 ROR
112108-01-7 | Ecopipam ( SCH 39166 )
(Catalog# : 25065)
Ecopipam (SCH 39166) 是一种有效的、选择性、具有口服活性的多巴胺