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Bromides
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Deuterated
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Indoles and Oxindoles
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
PROTAC
Antibody-drug Conjugate/ADC Related
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
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Piperidines
Pyridines
Pyrimidines
Quinolines
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Cas号索引 1
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Cas号索引 1
1314890-29-3 | TMP269
(Catalog# : 185254)
TMP269是一种具有高强度、选择性和可渗透性的IIa型HDAC抑制剂,其
1374743-00-6 | Trilaciclib (G1T28)
(Catalog# : 185235)
Trilaciclib是一种小分子竞争性细胞周期蛋白依赖性激酶4和6(CDK4 /
171235-71-5 | TAPI-1
(Catalog# : 185181)
TAPI-1是TACE的抑制剂。它抑制TNF-a、TNFRI(p60)和TNFRII(p80)的裂解。
158899-10-6 | TLN-232
(Catalog# : 18594)
TLN-232, 也称为CAP-232,是一种具有潜在抗肿瘤活性的合成环七肽。
140194-24-7 | 醋酸曲普瑞林
(Catalog# : 18592)
醋酸曲普瑞林是一种促性腺激素释放激素激动剂(GnRH激动剂),用作
1383816-29-2 | Tropifexor
(Catalog# : 18591)
Tropifexor, 也称为LJN452, 是一种用于治疗胆静性肝病和非酒精性脂肪
1702809-17-3 | THZ531
(Catalog# : 184172)
THZ531是一种共价CDK12和CDK13共价抑制剂。环素依赖性激酶12和13 (CDK
1802220-02-5 | TPX-0005
(Catalog# : 18423)
TPX-0005是一种Src/FAK/Janus激酶2 (JAK2)抑制剂。TPX-0005 + EGFR TKI抑制RTKs
1402601-82-4 | TUG-770
(Catalog# : 1791519)
TUG-770是高度有效的游离脂肪酸受体1(FFA1/GPR40)治疗2型糖尿病的激动
1429749-41-6 | Thiomyristoyl
(Catalog# : 1791113)
Thiomyristoyl是一种强效和特异性的IC50为28nM的SIRT2抑制剂。IC50与目标
1029877-94-8 | 琥珀酸曲格列汀
(Catalog# : 179811)
曲格列汀,也称为SYR472,是一种武田制药正在开发的治疗2型糖尿
1374516-07-0 | TUG-891
(Catalog# : 1783014)
TUG-891是一种有效且选择性的游离脂肪酸受体4(FFA4 / GPR120),它既显
1361951-15-6 | TP-3654
(Catalog# : 178303)
TP-3654是一种Pim-1和Pim-3激酶抑制剂,可用于治疗前列腺癌、急性髓
1326712-16-6 | TAK1抑制剂
(Catalog# : 1791412)
TAK1 inhibitor isis discontinued.TAK1抑制剂是一种有效的、相对选择性的
1351636-18-4 | Tirabrutinib游离 ( ONO-4059 )
(Catalog# : 17031303)
Tirabrutinib,也被称为ONO- 4059,是在抑制剂中,一种强大的、具有口
1610882-30-8 | TCS-OX2-29盐酸盐
(Catalog# : 17031302)
TCS-OX2- 29或TCS OX2 29,也被称为TCSOX229和TCS - OX229,是一种选择性的
1603845-32-4 | TX1-85-1
(Catalog# : 17030713)
TX1-85-1是一种ErbB3抑制剂. TX2-121-1可能通过异位机制发挥Her3依赖性
183204-72-0 | Tipiracil HCl
(Catalog# : 17030710)
Tipiralacil,又称TPI,是胸腺嘧啶磷酸化酶抑制剂(TPI)。Tipiracil是TAS
1234365-97-9 | Tenapanor HCl
(Catalog# : 17030113)
Tenapanor, 也称为AZD-1722和RDX 5791, 是钠-质子(Na(+)/ H(+))交换器NHE3的抑
150915-40-5 | 盐酸替罗非班
(Catalog# : 17030103)
替罗非班是一种抗血小板药物。它属于一种名为糖蛋白IIb / IIIa抑
135598-68-4 | TAS-109
(Catalog# : 17022810)
TAS-109, 也称为DFP-10917和CNDAC,是一种具有潜在抗肿瘤活性的核苷酸脱
1256037-58-7 | TRX818
(Catalog# : 17022401)
TRX-818是一种可口服的生物制剂,具有潜在的抗肿瘤活性和抗血管
15421-84-8 | 乐可安
(Catalog# : 17021310)
乐可安是一种PDGF拮抗剂,可抑制PDGF生成胶质瘤细胞的增殖。
1439901-97-9 | ONO-4059盐酸盐
(Catalog# : 17012103)
ONO-4059是BTK的选择性和新型抑制剂,IC50为2.2 nm,ONO-4059与B细胞内的
113942-30-6 | 替莫唑胺酸
(Catalog# : 17011905)
替莫唑胺酸, 也称为TMZA, 是一种具有明显抗癌活性的替奥米特(TMZ)
1609960-31-7 | TH588
(Catalog# : 17011728)
TH588是NUDT1的一种有效抑制剂,其IC50值为5nm,具有良好的代谢稳定
1415716-58-3 | TG6-10-1
(Catalog# : 17011727)
TG6-10-1是前列腺素E2受体亚型EP2的有效和选择性拮抗剂。
1033805-22-9 | 特罗司他乙酯
(Catalog# : 17011722)
特罗司他乙酯, 也称为LX 1032或LX 1606, 是一种口服血清素合成抑制剂
161715-24-8 | 泰比培南酯
(Catalog# : 17011721)
泰比培南酯,也被称为ME1211和TBM-PI, 是一种新型口腔卡宾枪抗生素。
193620-69-8 | TAS-301
(Catalog# : 17011719)
TAS-301是一种有效的、选择性的球囊冠状动脉过度拉伸损伤后的收
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
-- PROTAC
----
Molecular Glues
--
Antibody-drug Conjugate/ADC Related
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2763252-25-9 | M3554
(Catalog# : 25017)
M3554,一种新型抗GD2抗体药物偶联物。
| MD-43
(Catalog# : 25016)
MD-43是MCT4的强效选择性降解剂。
3034880-93-5 | VVD-130037 ( BAY-3605349 )
(Catalog# : 24110)
VVD-130037 (BAY-3605349) 是一种口服小分子 KEAP1 (INrf2) 激活剂。
2247396-91-2 | HC-5404 抑制剂
(Catalog# : 25001)
HC-5404 是一种新型、高选择性、有效的PERK抑制剂。
3034479-99-4 | HC-5404-FU
(Catalog# : 24112)
HC-5404-FU 是一种新型、高选择性、有效的PERK抑制剂。
2309409-79-6 | CMP-5 2HCl
(Catalog# : 24161)
CMP-5 is a potent, specific, and selective PRMT5 inhibitor, while displays no activit
2630378-05-9 | Wu-5
(Catalog# : 24160)
Wu-5 is a USP10 inhibitor that can inhibit FLT3 and AMPK pathways, induce FLT3-ITD de
890764-36-0 | VU-29
(Catalog# : 24159)
VU 29 is a potent allosteric potentiator at the rat mGlu5 receptor (EC50 = 9 nM); bin
1221186-52-2 | ML-202
(Catalog# : 24158)
ML-202 is an activator of pyruvate kinase M2 (PKM2).
921193-28-4 | BTA-EG4 hydrate
(Catalog# : 24157)
BTA-EG4 is a catalase-amyloid interaction inhibitor, which can significantly enhance