武汉永璨生物科技有限公司
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Indoles and Oxindoles
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
PROTAC
Antibody-drug Conjugate/ADC Related
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
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订购信息
联系我们
公司简介
联系我们
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产品名字索引 B
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产品名字索引 B
BAY-1436032
(Catalog# : 181181, Cas# :
1803274-65-8
)
BAY-1436032是一个强有力的,有选择性的,有效的突变异柠檬酸脱氢酶
BGB-283
(Catalog# : 17101620, Cas# :
1446090-77-2;1446090-79-4
)
BGB-283,也称为Beigene-283或Lifirafenib,是一种新的有效的和选择性的
Belizatinib
(Catalog# : 17101619, Cas# :
1357920-84-3
)
Belizatinib,也称为TSR-011,具有受体酪氨酸激酶间变性淋巴瘤激酶(
Bioymifi
(Catalog# : 1710165, Cas# :
1420071-30-2
)
Bioymifi是DR5的活性剂(Kd = 1.2 µM; IC50 = 2 µM). Bioymifi诱导凋亡的肿瘤
BLU-554
(Catalog# : 1710162, Cas# :
1707289-21-1
)
BLU-554是针对肝癌治疗的成纤维细胞生长因子受体4(FGFR4)抑制剂
BX-517
(Catalog# : 1791314, Cas# :
850717-64-5
)
BX-517,又名PDK1 inhibitor2,是强有力的和有选择性的PDK1抑制剂。
BBT-594
(Catalog# : 179133, Cas# :
882405-89-2
)
BBT594,也称为NVP-BBT594,是强有力的和有选择性的RET和JAK2抑制剂。
BAY41-4109消旋体
(Catalog# : 1791117, Cas# :
298708-79-9
)
Bay41-4109消旋体是对Bay41-4109和S-异构体Bay41-4109 R-异构体的混合物。
BAR-501
(Catalog# : 179821, Cas# :
1632118-69-4
)
BAR-501是一种选择性GPBAR1激动剂,没有任何的FXR激动剂活性。BAR-50
Batefenterol(free base)
(Catalog# : 179820, Cas# :
743461-65-6
)
Batefenterol,也称为 GSK961081和TD-5959,是一种毒蕈碱拮抗剂和β2-受体
BI-847325
(Catalog# : 83101, Cas# :
1207293-36-4
)
BI-847325是一种口服、具有选择性的日常生物MEK/Aurora激酶抑制剂,
BAY-598
(Catalog# : 17982, Cas# :
1906919-67-2
)
BAY-598是一种强效的针对SMYD2中肽-竞争的化学探测器。BAY-598拥有一
BAY-598 R-异构体
(Catalog# : 17981, Cas# :
1906920-28-2
)
BAY-598 R-异构体是BAY589 R-异构体。bay-598 R-异构体可以作为一个参照
布索芬新
(Catalog# : 17916, Cas# :
171655-91-7
)
布索芬新是一种充分的单胺再摄取阻滞剂,已被开发用于治疗帕金
B02
(Catalog# : 1783013, Cas# :
1290541-46-6
)
B02,也叫RAD51 - in - 02,是一种RAD51抑制剂。B02能增强MM细胞的DOX敏
BLU-285
(Catalog# : 1781003, Cas# :
1703793-34-3
)
BLU-285是一种有效、具有选择性的抑制剂。
BAY-1895344
(Catalog# : 1781002, Cas# :
1876467-74-1
)
BAY-1895344是一种有效的、具有选择性的ATM抑制剂。
BIBR1532
(Catalog# : 178813, Cas# :
321674-73-1
)
BIBR1132对端粒酶的抑制具有很强的选择性,导致肿瘤细胞延迟生长
BMS-932481
(Catalog# : 2017877, Cas# :
1263871-36-8
)
BMS-932481调节Aβ肽在血浆和脑脊液的健康志愿者。
B-1613
(Catalog# : 20178216, Cas# :
214066-78-1
)
(2S,4S)-4-(氨基甲基)吡咯烷-1,2-二羧酸 1-叔丁酯 2-甲酯;(2S,4S)-1-tert
Balamapimod
(Catalog# : 2017822, Cas# :
863029-99-6
)
<span style="color:#34495E;font-family:" font-Balamapimod, 也称为MKI-822,是一种
BP-1-102
(Catalog# : 17030606, Cas# :
1334493-07-0
)
BP-1-102是一种有效的口服生物和选择性抑制剂。
BAY-876
(Catalog# : 17030604, Cas# :
1799753-84-6
)
BAY-876是一种有效的、选择性的谷氨酸抑制剂。BAY- 876在体外具有良
BRD-7552
(Catalog# : 17030312, Cas# :
1137359-47-7
)
BRD-7552是一种PDX1转录诱导因子。它主要在人类胰岛和导管细胞中调
BDA-366
(Catalog# : 17030305, Cas# :
1821496-27-8
)
BDA - 366是BCL - BH4拮抗剂。BDA - 366抑制人骨髓瘤的生长。BDA - 366诱导
Bimiralisib
(Catalog# : 17030116, Cas# :
1225037-39-7
)
Bimiralisib,也被称为PQR309,是一种口服生物可用的磷脂- 3 -激酶抑
BEC HCl
(Catalog# : 17030110, Cas# :
222638-67-7
)
BEC,也称为S -(2-boronoethyl)-L-cysteine,是一个慢结合和竞争力的精氨酸
BGP-15
(Catalog# : 17109003, Cas# :
66611-37-8
)
BGP-15, 是一种带有PARP抑制活性的烟碱类胺肟衍生物。已经证明BGP-
Butylphthalide
(Catalog# : 16122908, Cas# :
6066-49-5
)
Butylphthalide, also known as 3-n-butylphthalide or NBP, is an antioxidant and one of
Buthionine Sulphoximine
(Catalog# : 16122907, Cas# :
5072-26-4
)
Buthionine Sulphoximine, also known as NSC-326231, is a gamma-glutamylcysteine synthe
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
-- PROTAC
----
Molecular Glues
--
Antibody-drug Conjugate/ADC Related
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
MGD-28
(Catalog# : 25073, Cas# :
2991818-13-2
)
MGD-28 is a potent molecular glue degrader that demonstrates significant in vitro eff
TG101209 analog 1
(Catalog# : 25072)
TG101209 analog 1 (Compound 8h) is an inhibitor of BUB1B with an IC50 of 10.36 μ M.
AT-007
(Catalog# : 25071, Cas# :
2170729-29-8
)
AT-007 is an orally active central nervous system (CNS) penetrant Aldose Reductase in
TAK-653
(Catalog# : 25070, Cas# :
1358751-06-0
)
TAK-653 is a novel AMPA receptor potentiator, strictly potentiating a glutamate-induc
Emavusertib
(Catalog# : 25069, Cas# :
1801344-14-8
)
Emavusertib, also known as CA-4948 is a potent IRAK4/FLT3 inhibitor with anti-tumor a
Roginolisib
(Catalog# : 25068, Cas# :
1305267-37-1
)
Roginolisib, also known as MSC2360844 and IOA-244, is a potent, orally active and sel
NT219
(Catalog# : 25067, Cas# :
1198078-60-2
)
NT219 is a novel inhibitor of the insulin/igf signaling cascade (iis), mediating a lo
SPB linker
(Catalog# : 25066, Cas# :
858128-57-1
)
SPB is a agent-linker conjugate for ADC with potent anti-inflammatory activity by usi
JTE-151
(Catalog# : 20594, Cas# :
1404380-58-0
)
JTE-151 是一种 RORγ 抑制剂,可通过抑制与 Th17 细胞活化相关的 ROR
Ecopipam ( SCH 39166 )
(Catalog# : 25065, Cas# :
112108-01-7
)
Ecopipam (SCH 39166) 是一种有效的、选择性、具有口服活性的多巴胺