武汉永璨生物科技有限公司
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others
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Aldehydes
Amines
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Anilines
Boronic Acids
Bromides
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Chiral Compounds
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Indoles and Oxindoles
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
PROTAC
Antibody-drug Conjugate/ADC Related
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
中间体
技术服务
定制合成
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订购信息
联系我们
公司简介
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产品名字索引 S
Seletalisib
(Catalog# : 1810221, Cas# :
1362850-20-1
)
Seletalisib,也被称为UCB-5857,是一种有效的选择性PI3激酶抑制剂,
Simenepag
(Catalog# : 1810172, Cas# :
910562-15-1
)
Simenepag,又名AGN-210676,是一种用于治疗青光眼和高眼压的小分子
SB-273005
(Catalog# : 186221, Cas# :
205678-31-5
)
SB-273005是一种整合素αvβ3的抑制剂。
STF-083010
(Catalog# : 185151, Cas# :
307543-71-1
)
STF-083010,也称为IRE1抑制剂I, 是IRE1/XBP1通路的抑制剂。
SAR407899游离
(Catalog# : 185115, Cas# :
923359-38-0
)
SAR407899是一种有效且具有选择性的、前景的抗高血压活性Rho激酶抑
SB-334867游离
(Catalog# : 185114, Cas# :
792173-99-0
)
SB-334867是一种阿立新拮抗剂。
SC-560
(Catalog# : 185113, Cas# :
188817-13-2
)
SC-560是一种有效的具有口服活性和选择性的COX-1抑制剂。
Seladelpar
(Catalog# : 185112, Cas# :
851528-79-5
)
Seladelpar,也被称为MBX-8025和RWJ-800025,是一种选择性的过氧化物酶
SEL120-34A盐酸盐
(Catalog# : 18574, Cas# :
1609452-30-3
)
SEL120-34A是一种高效、选择性的CDK8抑制剂,活跃于AML细胞中,具有
SR-4370
(Catalog# : 1842814, Cas# :
1816294-67-3
)
SR-4370是一种HDAC抑制剂。
SGC2085盐酸盐
(Catalog# : 184287, Cas# :
1821908-49-9
)
SGC2085是一种强效的选择性共激活剂,它可以使精氨酸甲基转移酶
S38093盐酸盐
(Catalog# : 184176, Cas# :
1222097-72-4
)
S38093是组胺H3受体的反向激动剂。
STO-609醋酸盐
(Catalog# : 184123, Cas# :
1173022-21-3
)
STO-609是一种细胞渗透性抑制剂,钙/钙调蛋白依赖性激酶激酶(CaMK
Super-TDU
(Catalog# : 18495, Cas# :
1599441-71-0
)
Super-TDU是靶向YAP-TEADs interaction的抑制性多肽。
SSD114 HCl
(Catalog# : 18427, Cas# :
N/A
)
SSD114是一种GABAB阳性变构调制器。SSD114增强gaba刺激[35S]GTP S与本地
(S)-(4-(3-(tert-butoxycarbonyl)-1-(isoquinolin-6-ylamino)-1-oxopropan-2-yl)phenyl)methyl 2,4-dimethylbenzoate
(Catalog# : 183219, Cas# :
1253955-19-9
)
(S)-(4-(3-(tert-butoxycarbonyl)-1-(isoquinolin-6-ylamino)-1-oxopropan-2-yl)phenyl)met
(S)-3-(tert-butoxycarbonyl)-2-(4-((2,4-dimethylbenzoyloxy)methyl)phenyl)propanoic acid
(Catalog# : 183218, Cas# :
2097334-20-6
)
(S)-3-(tert-butoxycarbonyl)-2-(4-((2,4-dimethylbenzoyloxy)methyl)phenyl)propanoic aci
(S)-2-羟基丁酸正丁酯
(Catalog# : 1712291, Cas# :
132513-51-0
)
(S)-2-羟基丁酸正丁酯是一种分子砌块。
SCR7 pyrazine
(Catalog# : 1712261, Cas# :
14892-97-8
)
SCR7吡嗪是DNA连接酶IV的小分子抑制剂,防止非同源端连接通过干扰
S38093
(Catalog# : 17101615, Cas# :
862896-30-8
)
S 38093 是一种大脑渗透的 H3 receptor 拮抗剂,对大鼠,小鼠和人的
SAR-7334盐酸
(Catalog# : 17101610, Cas# :
1333207-63-8
)
SAR-7334是一种新颖的、高效的、生物可利用的TRPC6通道,打开了新
SEN-826
(Catalog# : 1710168, Cas# :
1160833-51-1
)
SEN-826是一种潜在抗癌剂。
SRT3025 HCl
(Catalog# : 17101310, Cas# :
2070015-26-6
)
SRT3025是一种可口服的小分子激活SIRT1酶。
Senexin A
(Catalog# : 1710136, Cas# :
1366002-50-7
)
Senexin A是一种强效的选择性与抑制剂(IC50 = 280 nm)。Senexin A结合
S63845
(Catalog# : 171071, Cas# :
1799633-27-4
)
s63845是专门结合MCL1的BH3结合槽高亲和力的小分子。s63845有效杀死
Salermide
(Catalog# : 1791511, Cas# :
1105698-15-4
)
salermide是一个强大的肿瘤特异性凋亡的影响长寿基因蛋白质抑制剂
SD-06
(Catalog# : 1791320, Cas# :
271576-80-8
)
SD-06是治疗关节炎的MAPK p38α抑制剂。
Sulfatinib
(Catalog# : 179135, Cas# :
1308672-74-3
)
Sulfatinib是一种口服的血管内皮生长因子受体(VEGFR)1, 2,3,和成
S107 HCl
(Catalog# : 1791111, Cas# :
927871-76-9
)
S107是类型1 利阿诺定受体(RYR1)稳定剂;结合 RyR1提高calstabin-1亲
司美利特盐酸盐
(Catalog# : 179830, Cas# :
101526-62-9
)
司美利特,也称为CK-1752,是III类抗心律失常药。它是一种选择性
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
-- PROTAC
----
Molecular Glues
--
Antibody-drug Conjugate/ADC Related
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
MGD-28
(Catalog# : 25073, Cas# :
2991818-13-2
)
MGD-28 is a potent molecular glue degrader that demonstrates significant in vitro eff
TG101209 analog 1
(Catalog# : 25072)
TG101209 analog 1 (Compound 8h) is an inhibitor of BUB1B with an IC50 of 10.36 μ M.
AT-007
(Catalog# : 25071, Cas# :
2170729-29-8
)
AT-007 is an orally active central nervous system (CNS) penetrant Aldose Reductase in
TAK-653
(Catalog# : 25070, Cas# :
1358751-06-0
)
TAK-653 is a novel AMPA receptor potentiator, strictly potentiating a glutamate-induc
Emavusertib
(Catalog# : 25069, Cas# :
1801344-14-8
)
Emavusertib, also known as CA-4948 is a potent IRAK4/FLT3 inhibitor with anti-tumor a
Roginolisib
(Catalog# : 25068, Cas# :
1305267-37-1
)
Roginolisib, also known as MSC2360844 and IOA-244, is a potent, orally active and sel
NT219
(Catalog# : 25067, Cas# :
1198078-60-2
)
NT219 is a novel inhibitor of the insulin/igf signaling cascade (iis), mediating a lo
SPB linker
(Catalog# : 25066, Cas# :
858128-57-1
)
SPB is a agent-linker conjugate for ADC with potent anti-inflammatory activity by usi
JTE-151
(Catalog# : 20594, Cas# :
1404380-58-0
)
JTE-151 是一种 RORγ 抑制剂,可通过抑制与 Th17 细胞活化相关的 ROR
Ecopipam ( SCH 39166 )
(Catalog# : 25065, Cas# :
112108-01-7
)
Ecopipam (SCH 39166) 是一种有效的、选择性、具有口服活性的多巴胺