武汉永璨生物科技有限公司
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others
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Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
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Pyridines
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Quinolines
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
PROTAC
Antibody-drug Conjugate/ADC Related
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
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产品名字索引 T
TWS-119
(Catalog# : 17030204, Cas# :
601514-19-6
)
TWS-119 是一种强有力的和糖原合酶选择性抑制剂激酶-3β(IC50 = 30 nM
Tenapanor HCl
(Catalog# : 17030113, Cas# :
1234365-97-9
)
Tenapanor, 也称为AZD-1722和RDX 5791, 是钠-质子(Na(+)/ H(+))交换器NHE3的抑
盐酸替罗非班
(Catalog# : 17030103, Cas# :
150915-40-5
)
替罗非班是一种抗血小板药物。它属于一种名为糖蛋白IIb / IIIa抑
TAS-109
(Catalog# : 17022810, Cas# :
135598-68-4
)
TAS-109, 也称为DFP-10917和CNDAC,是一种具有潜在抗肿瘤活性的核苷酸脱
TRX818
(Catalog# : 17022401, Cas# :
1256037-58-7
)
TRX-818是一种可口服的生物制剂,具有潜在的抗肿瘤活性和抗血管
乐可安
(Catalog# : 17021310, Cas# :
15421-84-8
)
乐可安是一种PDGF拮抗剂,可抑制PDGF生成胶质瘤细胞的增殖。
ONO-4059盐酸盐
(Catalog# : 17012103, Cas# :
1439901-97-9
)
ONO-4059是BTK的选择性和新型抑制剂,IC50为2.2 nm,ONO-4059与B细胞内的
替莫唑胺酸
(Catalog# : 17011905, Cas# :
113942-30-6
)
替莫唑胺酸, 也称为TMZA, 是一种具有明显抗癌活性的替奥米特(TMZ)
泰地罗新
(Catalog# : 17011904, Cas# :
328898-40-4
)
泰地罗新 (TIP) 是一种新型十六环的巨环,用于治疗牛和猪呼吸系
TH588
(Catalog# : 17011728, Cas# :
1609960-31-7
)
TH588是NUDT1的一种有效抑制剂,其IC50值为5nm,具有良好的代谢稳定
TG6-10-1
(Catalog# : 17011727, Cas# :
1415716-58-3
)
TG6-10-1是前列腺素E2受体亚型EP2的有效和选择性拮抗剂。
TG101209
(Catalog# : 17011726, Cas# :
936091-14-4
)
TG101209是一种新型的、有效的JAK2抑制剂,在多种多发性骨髓瘤(MM)
替尼泊甙
(Catalog# : 17011723, Cas# :
29767-20-2
)
替尼泊甙是一种具有抗肿瘤活性的足叶草毒素的半合成衍生物。
特罗司他乙酯
(Catalog# : 17011722, Cas# :
1033805-22-9
)
特罗司他乙酯, 也称为LX 1032或LX 1606, 是一种口服血清素合成抑制剂
泰比培南酯
(Catalog# : 17011721, Cas# :
161715-24-8
)
泰比培南酯,也被称为ME1211和TBM-PI, 是一种新型口腔卡宾枪抗生素。
TC-H 106
(Catalog# : 17011720, Cas# :
937039-45-7
)
TC-H 106, 也称为Pimelic Diphenylamide 106, 是一种一类HDAC抑制剂,对II类
TAS-301
(Catalog# : 17011719, Cas# :
193620-69-8
)
TAS-301是一种有效的、选择性的球囊冠状动脉过度拉伸损伤后的收
TAS-103
(Catalog# : 17011718, Cas# :
174634-08-3
)
TAS-103,也称为BMS-247615, 是一种喹啉衍生物,在小鼠和人体肿瘤模型
Talabostat甲磺酸盐
(Catalog# : 17011717, Cas# :
150080-09-4
)
Talabostat, 也称为PT-100,具有抗肿瘤和造血作用的二肽肽酶抑制剂。
TAK-659盐酸盐
(Catalog# : 17011716, Cas# :
1312691-41-0
)
TAK-659是脾脏酪氨酸激酶(syk)的抑制剂,具有潜在的抗炎、免疫和抗
TAK-285
(Catalog# : 17011715, Cas# :
871026-44-7
)
TAK-285是一种新的双erbB蛋白激酶抑制剂,专门针对人类表皮生长因
盐酸坦索罗辛
(Catalog# : 17109008, Cas# :
106463-17-6
)
盐酸坦索罗辛是一个强有力的和选择性α1a肾上腺素能受体拮抗剂
T-0901317
(Catalog# : 16122840, Cas# :
293754-55-9
)
T-0901317, also known as T-1317; TO-091317; TO 901317, is a liver X receptor (LXR) ag
Terazosin
(Catalog# : 16122728, Cas# :
63074-08-8
)
Terazosin is a selective alpha-1 antagonist used for treatment of symptoms of an enla
Tubercidin
(Catalog# : 16122718, Cas# :
69-33-0
)
Tubercidin, an adenosine analogue, is a nucleoside antibiotic. It is incorporated int
TPO agonist 1
(Catalog# : 6111515, Cas# :
1033040-23-1
)
TPO agonist 1 can increase production of platelets by stimulating the TPO receptor in
TY-52156
(Catalog# : 61118, Cas# :
934369-14-9
)
TY-52156 is a potent S1P3 receptor antagonist in a competitive manner, and the Ki val
TCS-OX2-29
(Catalog# : 61117, Cas# :
372523-75-6
)
TCS-OX2-29 is a potent and selective OX2 receptor antagonist with IC50 of 40 nM. Disp
THZ1
(Catalog# : 6111013, Cas# :
1604810-83-4
)
THZ1 is a novel selective and potent covalent CDK7 inhibitor with IC50(binding affini
TZ9
(Catalog# : 611934, Cas# :
1002789-86-7
)
TZ9 is a novel inhibitor of Rad6 ubiquitin conjugating enzyme(E2 enzyme); inhibits MD
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
-- PROTAC
----
Molecular Glues
--
Antibody-drug Conjugate/ADC Related
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
MGD-28
(Catalog# : 25073, Cas# :
2991818-13-2
)
MGD-28 is a potent molecular glue degrader that demonstrates significant in vitro eff
TG101209 analog 1
(Catalog# : 25072)
TG101209 analog 1 (Compound 8h) is an inhibitor of BUB1B with an IC50 of 10.36 μ M.
AT-007
(Catalog# : 25071, Cas# :
2170729-29-8
)
AT-007 is an orally active central nervous system (CNS) penetrant Aldose Reductase in
TAK-653
(Catalog# : 25070, Cas# :
1358751-06-0
)
TAK-653 is a novel AMPA receptor potentiator, strictly potentiating a glutamate-induc
Emavusertib
(Catalog# : 25069, Cas# :
1801344-14-8
)
Emavusertib, also known as CA-4948 is a potent IRAK4/FLT3 inhibitor with anti-tumor a
Roginolisib
(Catalog# : 25068, Cas# :
1305267-37-1
)
Roginolisib, also known as MSC2360844 and IOA-244, is a potent, orally active and sel
NT219
(Catalog# : 25067, Cas# :
1198078-60-2
)
NT219 is a novel inhibitor of the insulin/igf signaling cascade (iis), mediating a lo
SPB linker
(Catalog# : 25066, Cas# :
858128-57-1
)
SPB is a agent-linker conjugate for ADC with potent anti-inflammatory activity by usi
JTE-151
(Catalog# : 20594, Cas# :
1404380-58-0
)
JTE-151 是一种 RORγ 抑制剂,可通过抑制与 Th17 细胞活化相关的 ROR
Ecopipam ( SCH 39166 )
(Catalog# : 25065, Cas# :
112108-01-7
)
Ecopipam (SCH 39166) 是一种有效的、选择性、具有口服活性的多巴胺