武汉永璨生物科技有限公司
+86-17702719238
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抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
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Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
PROTAC
Antibody-drug Conjugate/ADC Related
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
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Pyridines
Pyrimidines
Quinolines
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
PROTAC
Antibody-drug Conjugate/ADC Related
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
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产品名字索引 M
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产品名字索引 M
MBX-4132
(Catalog# : 2051511, Cas# :
2286411-30-9
)
MBX-4132 inhibit trans translation by binding to the bacterial ribosome.
ML188
(Catalog# : 2051506, Cas# :
1417700-13-0
)
ML188 is a Potent Noncovalent Small Molecule Inhibitor of the Severe Acute Respirator
ML277
(Catalog# : 2051504, Cas# :
1401242-74-7
)
ML277 is a potent activator of KCNQ1 (Kv7.1) channels with >100-fold selectivity v
4-(2-乙氨基)苯甲酸甲酯盐酸盐
(Catalog# : S-204149, Cas# :
56161-89-8
)
3-甲氧基-1-甲基-4-硝基-1H-吡唑
(Catalog# : 523192, Cas# :
1201935-85-4
)
Sun-shine Chemical provides 3-methoxy-1-methyl-4-nitro-1H-pyrazole(CAS 1201935-85-4)
3-甲氧基-1H-吡唑
(Catalog# : 523191, Cas# :
215610-30-3
)
Sun-shine Chemical provides 3-methoxy-1H-pyrazole (CAS 215610-30-3) with high quality
3-甲氧基-4-硝基-1H-吡唑
(Catalog# : 5141901, Cas# :
400755-41-1
)
methyl 2-bromo-5-fluoro-3-(4-methylphenylsulfonamido)benzoate
(Catalog# : 4281905, Cas# :
2086689-91-8
)
methyl 2-bromo-5-fluoro-3-(4-methylphenylsulfonamido)benzoate
MDK1846
(Catalog# : 193264, Cas# :
2102501-84-6
)
MDK1846是一种强效的酮己糖激酶(KHK)抑制剂。
MMG-11
(Catalog# : 1932010, Cas# :
313254-94-3
)
MMG-11是一种高效、选择性的TLR2/1和TLR2/6信号双抑制剂,具有较低的
ML221
(Catalog# : 19311, Cas# :
877636-42-5
)
ML221是apelin (APJ)受体的拮抗剂。
Melphalan flufenamide
(Catalog# : 192279, Cas# :
380449-51-4
)
Melphalan flufenamide,也称为前药J-1,是一种将烷基化剂美法仑与氟苯
ML184
(Catalog# : 192214, Cas# :
794572-10-4
)
ML184,也称为CID2440433,是一种有效的GPR55合成受体激动剂(EC50 = 0.26µM
Mitapivat
(Catalog# : 192191, Cas# :
1260075-17-9
)
Mitapivat,又称PKM2激活剂1020,是一种治疗丙酮酸激酶缺乏症的PKM2激
MK-3903
(Catalog# : 192183, Cas# :
1219737-12-8
)
MK-3903是一种有效的选择性AMPK激活剂(EC50 = 8 nM)。
Myriocin
(Catalog# : 191283, Cas# :
35891-70-4
)
多壳球菌素,又称抗生素ISP-1和热莫西丁,是一种非典型氨基酸,
MA242 TFA
(Catalog# : 191256, Cas# :
1049704-18-8
)
MA242是MDM2和NFAT1在胰腺癌治疗中的双重抑制剂。无论p53状态如何,
MIK665
(Catalog# : 191252, Cas# :
1799631-75-6
)
MIK665,又称s64315,诱导骨髓白血病细胞分化蛋白(mcl1;Bcl2-L-3),具有
MY 5445
(Catalog# : 191211, Cas# :
78351-75-4
)
MY 5445是一种潜在的血小板聚集抑制剂。
MRS1706
(Catalog# : 19131, Cas# :
264622-53-9
)
MRS1706是一种选择性腺苷A2B受体逆激动剂,人类A2B、A1、A2A、A3受体
MRS1177
(Catalog# : 1812296, Cas# :
183721-13-3
)
MRS1177是一种生物活性化学物。
MLN-4760
(Catalog# : 1812295, Cas# :
305335-31-3
)
MLN-4760是一种血管紧张素-转换(ACE2)抑制剂。在huMNCs中,MLN-4760-B检
MDK-8384
(Catalog# : 1812254, Cas# :
761438-38-4
)
MDK-8384,也称为ALK抑制剂2,是一种有效且具有选择性的ALK抑制剂。
Mavacamten
(Catalog# : 181255, Cas# :
1642288-47-8
)
Mavacamten,又称SAR-439152和MYK-461,是一种潜在的治疗肥厚性心肌病的
MK-2048
(Catalog# : 181251, Cas# :
869901-69-9
)
MK-2048是第二代HIV-1整合酶抑制剂。
ML 351
(Catalog# : 1811282, Cas# :
847163-28-4
)
ML 351是一种选择性的12/15 LOX抑制剂,在体内具有活性。
马罗皮坦
(Catalog# : 1811261, Cas# :
147116-67-4
)
马罗皮坦,又称CJ11972,是一种神经激肽(NK1)受体拮抗剂。
MBQ-167
(Catalog# : 181152, Cas# :
2097938-73-1
)
MBQ-167是一种有效的双Rac/Cdc42抑制剂,IC50分别为103/78 nM,用于转移
MDK4882
(Catalog# : 1810301, Cas# :
94164-88-2
)
MDK4882也称为PKM2抑制剂或化学物3k,是一种 PKM2抑制剂。
MU-380
(Catalog# : 181022, Cas# :
2109805-78-7
)
MU-380是一种有效且具有选择性的CHK1抑制剂。
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
-- PROTAC
----
Molecular Glues
--
Antibody-drug Conjugate/ADC Related
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
MGD-28
(Catalog# : 25073, Cas# :
2991818-13-2
)
MGD-28 is a potent molecular glue degrader that demonstrates significant in vitro eff
TG101209 analog 1
(Catalog# : 25072)
TG101209 analog 1 (Compound 8h) is an inhibitor of BUB1B with an IC50 of 10.36 μ M.
AT-007
(Catalog# : 25071, Cas# :
2170729-29-8
)
AT-007 is an orally active central nervous system (CNS) penetrant Aldose Reductase in
TAK-653
(Catalog# : 25070, Cas# :
1358751-06-0
)
TAK-653 is a novel AMPA receptor potentiator, strictly potentiating a glutamate-induc
Emavusertib
(Catalog# : 25069, Cas# :
1801344-14-8
)
Emavusertib, also known as CA-4948 is a potent IRAK4/FLT3 inhibitor with anti-tumor a
Roginolisib
(Catalog# : 25068, Cas# :
1305267-37-1
)
Roginolisib, also known as MSC2360844 and IOA-244, is a potent, orally active and sel
NT219
(Catalog# : 25067, Cas# :
1198078-60-2
)
NT219 is a novel inhibitor of the insulin/igf signaling cascade (iis), mediating a lo
SPB linker
(Catalog# : 25066, Cas# :
858128-57-1
)
SPB is a agent-linker conjugate for ADC with potent anti-inflammatory activity by usi
JTE-151
(Catalog# : 20594, Cas# :
1404380-58-0
)
JTE-151 是一种 RORγ 抑制剂,可通过抑制与 Th17 细胞活化相关的 ROR
Ecopipam ( SCH 39166 )
(Catalog# : 25065, Cas# :
112108-01-7
)
Ecopipam (SCH 39166) 是一种有效的、选择性、具有口服活性的多巴胺