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Name Index A

• AMG232 (Catalog# : 011911, Cas# : 1352066-68-2)AMG232 is an extremely potent MDM2 inhibitor (SPR KD = 0.045 nM, SJSA-1 EdU IC50 = 9.
• Afdx 384 (Catalog# : 011905, Cas# : 118290-27-0)Coming soon!
• Avoralstat (Catalog# : 011813, Cas# : 918407-35-9)Avoralstat (formerly BCX4161) is a potent small-molecule oral plasma kallikrein inhib
• AMG-337 (Catalog# : 01181, Cas# : 1173699-31-4)AMG-337 is a potent and highly selective small molecule ATP-competitive MET kinase in
• Afuresertib (Catalog# : 011811, Cas# : 1047644-62-1)Afuresertib is a potent pan-AKT inhibitor that demonstrated synergy with bortezomib i
• AMG 900 (Catalog# : 011803, Cas# : 945595-80-2)AMG 900 is a potent and highly selective pan-Aurora kinases inhibitor for Aurora A/B/
• APTO-253 (Catalog# : 011802, Cas# : 1422731-37-0)APTO-253 is a small molecule inhibitor of human metal-regulatory transcription factor
• AC-55541 (Catalog# : 011302, Cas# : 916170-19-9)AC-55541 is a novel small-molecule protease-activated receptor 2(PAR2) agonist.
• AZ 628 (Catalog# : 011120, Cas# : 878739-06-1)AZ628 is a new pan-Raf inhibitor for BRAF, BRAFV600E, and c-Raf-1 with IC50 of 105 nM
• AZD-5582 (Catalog# : 011117, Cas# : 1258392-53-8)AZD5582 is a potent IAP inhibitor, which is a dimeric compound based on the AVPI moti
• Arbidol hydrochloride (Catalog# : 011111, Cas# : 131707-23-8)Arbidol is an broad-spectrum antiviral chemical agent which can inhibit cell entry of
• APY29 (Catalog# : 011108, Cas# : 1216665-49-4)APY29 is an allosteric modulator of IRE1; inhibits IRE1 autophosphorylation (IC50 = 2
• AMG-47a (Catalog# : 011107, Cas# : 882663-88-9)AMG-47a is a potent inhibitor of Lck and T cell proliferation.
• ARQ-736 (Catalog# : 011104, Cas# : 1228237-57-7)ARQ 736 is a potent and selective BRAF inhibitor.
• AZD4547 (Catalog# : 010820, Cas# : 1035270-39-3)AZD4547 is a novel selective FGFR inhibitor targeting FGFR1/2/3 with IC50 of 0.2 nM/2
• AZD-1480 (Catalog# : 010816, Cas# : 935666-88-9)AZD1480 is a novel ATP-competitive JAK2 inhibitor with IC50 of 0.26 nM, selectivity a
• AZD8330 (Catalog# : 010809, Cas# : 869357-68-6)AZD8330 is a novel, selective, non-ATP competitive MEK 1/2 inhibitor with IC50 of 7 n
• AS703026 (Catalog# : 010808, Cas# : 1236699-92-5)AS703026 is an orally bioavailable small-molecule inhibitor of MEK1 and MEK2 (MEK1/2)
• AZ505 (Catalog# : 010803, Cas# : 1035227-43-0)AZ505 is a potent and highly selective inhibitor of the oncogenic protein SMYD2(IC50=
• AG-L-59687 (Catalog# : 010428, Cas# : 793035-88-8)Coming soon!
• AG1024 (Catalog# : 010422, Cas# : 65678-07-1)AG-1024 inhibits IGF-1R autophosphorylation with IC50 of 7 M, less potent to IR with
• Almotriptan (Catalog# : 010418, Cas# : 154323-57-6)Almotriptan is a 5-HT1B/1D-receptor agonist used to treat migraine.
• AM630 (Catalog# : 010410, Cas# : 164178-33-0)AM630 is a selectivity CB2 antagonist with Ki of 31.2 nM; > 150 fold selectivity o
• AZD-8055 (Catalog# : 123019, Cas# : 1009298-09-2)AZD-8055 is an inhibitor of the mammalian target of rapamycin (mTOR) with potential a
• Amuvatinib (Catalog# : 123016, Cas# : 850879-09-3)Amuvatinib is a potent and multi-targeted inhibitor of c-Kit, PDGFR and Flt3 with IC5
• AR-42 (Catalog# : 123009, Cas# : 935881-37-1)AR-42 is a novel, oral cancer therapy currently in early clinical development.
• A-966492 (Catalog# : 123006, Cas# : 934162-61-5)A-966492 is a novel and potent inhibitor of PARP1 and PARP2 with Ki of 1 nM and 1.5 n
• AMG 487 (Catalog# : 122942, Cas# : 473719-41-4)AMG 487 is a small molecule antagonist of the chemokine receptor CXCR3.
• Atosiban acetate (Catalog# : 122931, Cas# : 90779-69-4)Atosiban is a nonapeptide, desamino-oxytocin analogue, and a competitive vasopressin/
• AST-1306 (Catalog# : 122926, Cas# : 897383-62-9)AST-1306 is a novel irreversible inhibitor of EGFR and ErbB2 with IC50 of 0.5 nM and